1: With n-butyllithium in tetrahydrofuran T=-78°C; 0.25 h; 2: With boric acid trimethyl ester in tetrahydrofuran T=20°C; 1 h; 3: With hydrogenchloride; water in tetrahydrofuran
参考文献
Raje, Mithun R.; Knott, Kenneth; Kharel, Yugesh; Bissel, Philippe; Lynch, Kevin R.; Santos, Webster L.
Bioorganic and Medicinal Chemistry, 2012 , vol. 20, # 1 p. 183 - 194