1: With water; potassium hydroxide in ethanol
1 h; Reflux;
2: With hydrogenchloride in ethanol; water
参考文献
GLAXO GROUP LIMITED; CHONG, Pek Yoke; MILLER, John F.; PEAT, Andrew James; SHOTWELL, John Brad
Patent: WO2013/28371 A1, 2013 ;
Location in patent: Page/Page column 36 ;