1.1: triphenylphosphine / tetrahydrofuran / 0.17 h / 20 °C 1.2: 0.67 h / 20 °C 2.1: hydrogenchloride; water / dichloromethane / 18 h / 20 °C 2.2: 0.75 h / 20 °C / pH 7 - 8 View Scheme
参考文献
ALPHORA RESEARCH INC.; ALBERICO, Dino; CLAYTON, Joshua; DIXON, Craig; GORIN, Boris
Patent: WO2011/150512 A1, 2011 ;
1.1: triphenylphosphine / tetrahydrofuran / 0.17 h / 20 °C 1.2: 0.67 h / 20 °C 2.1: hydrogenchloride; water / dichloromethane / 18 h / 20 °C 2.2: 0.75 h / 20 °C / pH 7 - 8 View Scheme
参考文献
ALPHORA RESEARCH INC.; ALBERICO, Dino; CLAYTON, Joshua; DIXON, Craig; GORIN, Boris
Patent: WO2011/150512 A1, 2011 ;