反应条件
1: 94 percent / DMAP / CH2Cl2 / 1 h / 0 °C 2: 26 percent / K2CO3 / dimethylsulfoxide / 85 °C 3: 1) BBr3, 2) aq. NH3 / 1) CH2Cl2, 2) CH2Cl2, 45 min View Scheme
参考文献
Jones, Martin F.; Noble, Stewart A.; Robertson, Colin A.; Storer, Richard
Tetrahedron Letters, 1991 , vol. 32, # 2 p. 247 - 250