反应条件
1: sodium hydride / N,N-dimethyl-formamide / 1 h / 20 °C
2: potassium carbonate / N,N-dimethyl-formamide / 1.5 h / 70 °C
View Scheme
参考文献
Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Tabarrini, Oriana; Kaatz, Glenn W.; Patel, Diixa; Cecchetti, Violetta
Journal of Medicinal Chemistry, 2011 , vol. 54, # 16 p. 5722 - 5736