反应条件
1: 80 percent / pyridine / 0.75 h / Ambient temperature 2: 1.) 0.1 M phosphate buffer (pH=7.8), 2.) 7 N aq. HCl / 1.) 95percent aq. ethanol, 48 deg C, 2.5 h, 2.) reflux, 8 h View Scheme
参考文献
Elfarra; Hanna
Journal of Medicinal Chemistry, 1985 , vol. 28, # 10 p. 1453 - 1460