尼非卡兰中间体B4(1,3-二甲基-6-[2-(对甲基苯磺酰氧基)乙基胺]-2,4(1H.3H)-嘧啶双酮合成路线 (共 1 条)
反应条件
sodium hydroxide; toluene-4-sulfonic acid 1.) methanol, 50 deg C, 2.) 80 deg C, 1 h; Yield given. Multistep reaction;
参考文献
Katakami; Yokoyama; Miyamoto; Mori; Kawauchi; Nobori; San-nohe; Kaiho; Kamiya
Journal of Medicinal Chemistry, 1992 , vol. 35, # 18 p. 3325 - 3330