1-BOC-3,5-二甲基哌嗪合成路线 (共 3 条)
反应条件
in tetrahydrofuran T=20°C; 4 h;
参考文献
Zhang, Nan; Zhong, Rong
Patent: US2013/116265 A1, 2013 ;
Location in patent: Paragraph 0024; 0025 ;
反应条件
1: in dichloromethane T=0 - 20°C; 2: With potassium carbonate in dichloromethane; water
参考文献
US2009/264416 A1, ;
Page/Page column 32 ;
反应条件
sodium hydroxide in water
参考文献
WO2006/46031 A1, ;
Page/Page column 50-51 ;
WO 2006/046031 A1