3-(三氟甲基)-1H-吡唑-5-甲酰氯合成路线 (共 1 条)
反应条件
1: With lithium aluminium tetrahydride in tetrahydrofuran
T=20°C; 48 h;
2: With methanol in tetrahydrofuran
参考文献
N.V. ORGANON
Patent: WO2008/3452 A1, 2008 ;
Location in patent: Page/Page column 58-59 ;
WO 2008/003452 A1