反应条件
methanol; ammonia; sodium hydride 1.) DMF, RT, 3 days, 2.) 100 deg C, overnight; Yield given. Multistep reaction. Yields of byproduct given;
参考文献
Jie, Liu; Aerschot, Arthur Van; Balzarini, Jan; Janssen, Gerard; Busson, Roger; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 9 p. 2481 - 2487