1: oxalyl chloride, DMF / CH2Cl2 / 1 h 2: Et3N / CH2Cl2 / 2 h View Scheme
参考文献
Bermudez, Jose; Fake, Charles S.; Joiner, Graham F.; Joiner, Karen A.; King, Frank D.; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 7 p. 1924 - 1929
triethylamine in dichloromethane 2 h; Yield given;
参考文献
Bermudez, Jose; Fake, Charles S.; Joiner, Graham F.; Joiner, Karen A.; King, Frank D.; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 7 p. 1924 - 1929