1-N-Boc-4-苯胺基哌啶合成路线 (共 11 条)
反应条件
palladium diacetate; potassium tert-butylate; 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl in tetrahydrofuran; toluene
T=110°C; 16 h;
参考文献
Thoma, Gebhard; Nuninger, Francois; Schaefer, Marc; Akyel, Kayhan G.; Albert, Rainer; Beerli, Christian; Bruns, Christian; Francotte, Eric; Luyten, Marcel; MacKenzie, Duncan; Oberer, Lukas; Streiff, Markus B.; Wagner, Trixie; Walter, Hansrudolf; Weckbecker, Gisbert; Zerwes, Hans-Guenter
Journal of Medicinal Chemistry, 2004 , vol. 47, # 8 p. 1939 - 1955