反应条件
1: N-(3-(3-cyanopyrazolo[1,5-a]pyrimidin-5-yl)phenyl)acetamide With sodium hydride in N,N-dimethyl-formamide
T=20°C; 1 h;
2: ethyl iodide in N,N-dimethyl-formamide
T=20°C; 24 h;
参考文献
Radl, Stanislav; Blahovcova, Michaela; Tkadlecova, Marcela; Havlicek, Jaroslav
Heterocycles, 2010 , vol. 80, # 2 p. 1359 - 1376