反应条件
1: 60 percent / HBr, AcOH / CHCl3 / 20 h / Ambient temperature
2: 70 percent / ICl / acetic acid / 1.) reflux, 3 h, 2.) room temperature, 18 h
View Scheme
参考文献
Kung; Kasliwal; Pan; Mach; Guo
Journal of Medicinal Chemistry, 1988 , vol. 31, # 5 p. 1039 - 1043