反应条件
1: H2, AcOH / 10percent Pd/C / ethanol / 60 °C 2: K2CO3, KI / butan-2-one / 17 h / Heating 3: 10percent HCl / 4 h / Heating 4: 1-ethyl-3-<3-(dimethylamino)propyl>carbodiimide hydrochloride / CH2Cl2 / 4 h / Ambient temperature View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 34, # 2 p. 616 - 624