反应条件
1: molecular sieves 4A / toluene / 1 h / 0 °C 2: (R)-1,1'-binaphthyl-3,3'-bis(Ph2P=O)-2,2'-diyl-AlCl; PhOH / CH2Cl2 / 44 h / -40 °C 3: MnO2 / CH2Cl2 / 1 h / 20 °C 4: 1 N aq. HCl / tetrahydrofuran / 1 h / 20 °C 5: aq. HCl / 24 h / 120 °C View Scheme
参考文献
Chemical and Pharmaceutical Bulletin, , vol. 48, # 10 p. 1586 - 1592