呋喃并[3,2-c]吡啶-2-羧醛合成路线 （共 7 条）
反应条件
formic acid in water
参考文献
Wishka, Donn G.; Reitz, Steven Charles; Piotrowski, David W.; Groppi JR., Vincent E.
Patent: US2003/45540 A1, 2003 ;
反应条件
Yield given. Multistep reaction;
参考文献
Saari, Walfred S.; Wai, John S.; Fisher, Thorsten E.; Thomas, Craig M.; Hoffman, Jacob M.; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 21 p. 3792 - 3802
反应条件
1: 95 percent / hydroxylamine hydrochloride, K2CO3 / aq. ethanol / 2 h / Ambient temperature 2: 65 percent / p-toluenesulfonic acid, acetic anhydride / 5 h / Heating View Scheme
参考文献
Journal of Heterocyclic Chemistry, , vol. 24, p. 373 - 376
反应条件
potassium dihydrogenphosphate; NaClO2 in water; dimethyl sulfoxide
参考文献
Wishka, Donn G.; Reitz, Steven Charles; Piotrowski, David W.; Groppi JR., Vincent E.
Patent: US2003/45540 A1, 2003 ;
反应条件
1: AcOH / ethanol / Ambient temperature 2: NaCNBH3 / ethanol / 1 h / Ambient temperature View Scheme
参考文献
Saari, Walfred S.; Wai, John S.; Fisher, Thorsten E.; Thomas, Craig M.; Hoffman, Jacob M.; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 21 p. 3792 - 3802
反应条件
potassium hydroxide; hydrazine hydrate in ethanol 1 h; Heating;
参考文献
Morita, Hiroyuki; Shiotani, Shunsaku
Journal of Heterocyclic Chemistry, 1987 , vol. 24, p. 373 - 376
反应条件
1: With sodium tetrahydroborate in methanol
T=0°C; 1.5 h;
2: With water in methanol
参考文献
Prosidion Ltd
Patent: WO2006/67532 A1, 2006 ;
Location in patent: Page/Page column 19-20 ;
WO 2006/067532 A1
