1: With potassium carbonate; Pd-Tedicyp catalyst in N,N-dimethyl-formamide T=110°C; Heck reaction; 20 h; 2: With sodium hydroxide; water in N,N-dimethyl-formamide T=50 - 80°C;
参考文献
Lemhadri, Mhamed; Doucet, Henri; Santelli, Maurice
Tetrahedron, 2004 , vol. 60, # 50 p. 11533 - 11540
1: Pd(PPh3)4; LiCl; CuCl / 80 °C 2: H2 / PtO2 / ethanol / 20 °C View Scheme
参考文献
Lin, Peter; Parikh, Mamta; Lo, Jane-Ling; Yang, Yi Tien; Cheng, Kang; Smith, Roy G; Fisher, Michael H; Wyvratt, Matthew J; Goulet, Mark T
Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 8 p. 1077 - 1080
