反应条件
1: 1.) 1,1'-carbonyldiimidazole (CDI), 2.) Et3N / 1.) THF, a) 0 deg C 3 h, b) RT, 4 h, 2.) THF, CH3CN, RT, 16 h 2: 1,4-diazabicyclo<2.2.2>octane (DABCO) / xylene / 5 h / Heating View Scheme
参考文献
Augelli-Szafran; Blankley; Roth; Trivedi; Bousley; Essenburg; Hamelehle; Krause; Stanfield
Journal of Medicinal Chemistry, 1993 , vol. 36, # 20 p. 2943 - 2949
