反应条件
1: 64 percent / chlorobenzene / 9 h / 100 - 105 °C 2: 65 percent / tetrahydrofuran / 1.5 h / Ambient temperature 3: 76 percent / AlCl3, n-propanethiol / 1,2-dichloro-ethane / 5 h / 5 - 20 °C View Scheme
参考文献
Grese, Timothy A.; Cho, Stephen; Finley, Don R.; Godfrey, Alexander G.; Jones, Charles D.; Lugar III, Charles W.; Martin, Michael J.; Matsumoto, Ken; Pennington, Lewis D.; Winter, Mark A.; Adrian, M. Dee; Cole, Harlan W.; Magee, David E.; Phillips, D. Lynn; Rowley, Ellen R.; Short, Lorri L.; Glasebrook, Andrew L.; Bryant, Henry U.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 2 p. 146 - 167