反应条件
Multi-step reaction with 4 steps 1: Et3N / toluene / 3 h / Heating2: NaH / dimethylformamide3: B(OH)3, (EtO)3B / Heating4: 1.) Et3N, 2.) Et3N, water / 1.) diethyl ether, RT, 5 h, 2.) diethyl ether, reflux, 2 h
参考文献
Godfroid, Jean-Jacques; Broquet, Colette; Jouquey, Simone; Lebbar, Mariya; Heymans, Francoise; et al. Journal of Medicinal Chemistry, 1987 , vol. 30, # 5 p. 792 - 797
