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5-氨基-2-(三氟甲基)吡啶合成路线 (共 11 条)
参考文献
Journal of Heterocyclic Chemistry, , vol. 31, # 6 p. 1413 - 1416
参考文献
Pinard, Emmanuel; Alanine, Alexander; Alberati, Daniela; Bender, Markus; Borroni, Edilio; Bourdeaux, Patrick; Brom, Virginie; Burner, Serge; Fischer, Holger; Hainzl, Dominik; Halm, Remy; Hauser, Nicole; Jolidon, Synese; Lengyel, Judith; Marty, Hans-Peter; Meyer, Thierry; Moreau, Jean-Luc; Mory, Roland; Narquizian, Robert; Nettekoven, Mathias; Norcross, Roger D.; Puellmann, Bernd; Schmid, Philipp; Schmitt, Sebastien; Stalder, Henri; Wermuth, Roger; Wettstein, Joseph G.; Zimmerli, Daniel
Journal of Medicinal Chemistry, 2010 , vol. 53, # 12 p. 4603 - 4614
参考文献
Probst, Gary; Aubele, Danielle L.; Bowers, Simeon; Dressen, Darren; Garofalo, Albert W.; Hom, Roy K.; Konradi, Andrei W.; Marugg, Jennifer L.; Mattson, Matthew N.; Neitzel, Martin L.; Semko, Chris M.; Sham, Hing L.; Smith, Jenifer; Sun, Minghua; Truong, Anh P.; Ye, Xiaocong M.; Xu, Ying-Zi; Dappen, Michael S.; Jagodzinski, Jacek J.; Keim, Pamela S.; Peterson, Brian; Latimer, Lee H.; Quincy, David; Wu, Jing; Goldbach, Erich; Ness, Daniel K.; Quinn, Kevin P.; Sauer, John-Michael; Wong, Karina; Zhang, Hongbin; Zmolek, Wes; Brigham, Elizabeth F.; Kholodenko, Dora; Hu, Kang; Kwong, Grace T.; Lee, Michael; Liao, Anna; Motter, Ruth N.; Sacayon, Patricia; Santiago, Pamela; Willits, Christopher; Bard, Frederique; Bova, Michael P.; Hemphill, Susanna S.; Nguyen, Lam; Ruslim, Lany; Tanaka, Kevin; Tanaka, Pearl; Wallace, William; Yednock, Ted A.; Basi, Guriqbal S.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 13 p. 5261 - 5274
参考文献
ASTRAZENECA AB
Patent: WO2006/4533 A1, 2006 ;
Location in patent: Page/Page column 25 ;
WO 2006/004533 A1
参考文献
NOVARTIS AG
Patent: WO2009/50183 A2, 2009 ;
Location in patent: Page/Page column 121 ;
参考文献
AMGEN INC.
Patent: WO2009/51718 A2, 2009 ;
Location in patent: Page/Page column 45 ;
WO 2009/051718 A2
参考文献
IRM LLC; CORTEZ, Alex; LI, Yongkai; LIAO, Xuebin; WU, Tom Yao-Hsiang; ZHANG, Xiaoyue
Patent: WO2011/57148 A1, 2011 ;
Location in patent: Page/Page column 102 ;
参考文献
Almirall, S.A.; Vidal Juan, Bernat; Alonso Diez, Juan Antonio; Buil Albero, María Antonia; Eastwood, Paul Robert; Esteve Trias, Cristina; Lozoya Toribio, María Estrella; Roberts, Richard Spurring; Vidal Gispert, Laura
Patent: EP2548876 A1, 2013 ;
Location in patent: Paragraph 0333-0336 ;
EP 2548876 A1
参考文献
Almirall, S.A.; Vidal Juan, Bernat; Alonso Diez, Juan Antonio; Buil Albero, María Antonia; Eastwood, Paul Robert; Esteve Trias, Cristina; Lozoya Toribio, María Estrella; Roberts, Richard Spurring; Vidal Gispert, Laura
Patent: EP2548876 A1, 2013 ;
EP 2548876 A1
参考文献
Swanson, Devin M.; Dubin, Adrienne E.; Shah, Chandra; Nasser, Nadia; Chang, Leon; Dax, Scott L.; Jetter, Michele; Breitenbucher, J. Guy; Liu, Changlu; Mazur, Curt; Lord, Brian; Gonzales, Lisa; Hoey, Kenway; Rizzolio, Michele; Bogenstaetter, Michael; Codd, Ellen E.; Lee, Doo H.; Zhang, Sui-Po; Chaplan, Sandra R.; Carruthers, Nicholas I.
Journal of Medicinal Chemistry, 2005 , vol. 48, # 6 p. 1857 - 1872
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