反应条件
1: 95 percent / dicyclohexylcarbodiimide (DCC), 1-hydroxybenzotriazole (HOBT), Et3N / dimethylformamide / 144 h / 5 °C 2: ethanol / 18 h / 20 °C View Scheme
参考文献
McElroy, Andrew B.; Clegg, Stephen P.; Deal, Martyn J.; Ewan, Georg B.; Hagan, Russell M.; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 14 p. 2582 - 2591
