反应条件
1: H2SO4 2: 82 percent / aq. NaBH4 / methanol / 2 h / Heating 3: 80 percent / pyridine / 3 h / Ambient temperature 4: 1.) NaH / 1.) DMF, 2.) DMF, 90 deg C, 2 h View Scheme
参考文献
Ohno; Adachi; Koumori; Mizukoshi; Nagasaka; Ichihara; Kato -
Chemical and Pharmaceutical Bulletin, 1994 , vol. 42, # 7 p. 1463 - 1473