1: With potassium phosphate; trifluoromethyl amino ketone; N-methyl-2-(methylamino)ethylamine; copper(l) iodide in N,N-dimethyl-formamide T=45°C; 2: With methanol in N,N-dimethyl-formamide T=45°C; Further stages.;
1: With Zn[N(SiMe3)2]2; tri-tert-butyl phosphine; tetrabutylammomium bromide; bis(dibenzylideneacetone)-palladium(0) in tetrahydrofuran T=50°C; 24 h; 2: With hydrogenchloride in tetrahydrofuran; diethyl ether
参考文献
Lee, Dae-Yon; Hartwig, John F.
Organic Letters, 2005 , vol. 7, # 6 p. 1169 - 1172
