1: With n-butyllithium in tetrahydrofuran; hexane T=-78°C; 0.666667 h; 2: With boric acid trimethyl ester in tetrahydrofuran; hexane T=-78 - 20°C; 18 h; 3: With hydrogenchloride in tetrahydrofuran; hexane; water
参考文献
Bristol-Myers Squibb Company
Patent: US2007/3539 A1, 2007 ;
Location in patent: Page/Page column 71 ;
US 20070003539 A1