反应条件
1: With acetic acid in 1,2-dichloro-ethane
18 h;
2: With sodium tris(acetoxy)borohydride in 1,2-dichloro-ethane
1 h;
参考文献
Chiasson, Jean-Franois; Boulet, Louise; Brideau, Christine; Chau, Anh; Claveau, David; Cote, Bernard; Ethier, Diane; Giroux, Andre; Guay, Jocelyne; Guiral, Sebastien; Mancini, Joseph; Masse, Frederic; Methot, Nathalie; Riendeau, Denis; Roy, Patrick; Rubin, Joel; Xu, Daigen; Yu, Hongping; Ducharme, Yves; Friesen, Richard W.
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 5 p. 1488 - 1492