反应条件
1: potassium hydroxide; N-benzyl-N,N,N-triethylammonium chloride / toluene / 20 °C / |Inert atmosphere 2: anhydrous xylene / 48 h / 150 °C / |Inert atmosphere View Scheme
参考文献
GENENTECH, INC.; FORMA TM, LLC; BAIR, Kenneth, W.; BAUMEISTER, Timm, R.; GOSSELIN, Francis; ZAK, Mark; ZHENG, Xiaozhang
Patent: WO2013/130935 A1, 2013 ;
Title/Abstract Full Text Show Details
GENENTECH, INC.; FORMA TM, LLC; BAIR, Kenneth, W.; BAUMEISTER, Timm, R.; BUCKMELTER, Alexandre, J.; CLODFELTER, Karl, H.; GUNZNER-TOSTE, Janet; HAN, Bingsong; LIN, Jian; REYNOLDS, Dominic, J.; SMITH, Chase, C.; WANG, Zhongguo; ZAK, Mark; ZHENG, Xiaozhang; ZHAO, Guiling
Patent: WO2013/130943 A1, 2013 ;