反应条件
1.1: n-butyllithium / tetrahydrofuran / 1 h / -78 °C / |Inert atmosphere 1.2: 2 h / -78 °C / |Inert atmosphere 1.3: 5 h / 20 °C / |Inert atmosphere 2.1: methanol / 15 h / 20 °C / |Inert atmosphere 3.1: PdCl2dcpp; copper(l) iodide; 2-methylamino-ethanol / N,N-dimethyl-formamide / 16 h / 100 °C / |Inert atmosphere View Scheme
参考文献
Organic Letters, , vol. 15, # 17 p. 4308 - 4311