反应条件
1: With thionyl chloride; N,N-dimethyl-formamide in tetrahydrofuran T=10 - 25°C; 2: With hydrogenchloride; ammonia in tetrahydrofuran; water; N,N-dimethyl-formamide T=-10 - 30°C; 1 h;
参考文献
Engstrom, Kenneth M.; Baize, Amanda L.; Franczyk, Thaddeus S.; Kallemeyn, Jeffrey M.; Mulhern, Mathew M.; Rickert, Robert C.; Wagaw, Seble
Journal of Organic Chemistry, 2009 , vol. 74, # 10 p. 3849 - 3855